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Trial details imported from ClinicalTrials.gov

For full trial details, please see the original record at https://clinicaltrials.gov/study/NCT00710684




Registration number
NCT00710684
Ethics application status
Date submitted
30/06/2008
Date registered
4/07/2008
Date last updated
7/12/2017

Titles & IDs
Public title
A Study of SB-742457, Added to Donepezil for the Treatment of Mild-to-moderate Alzheimer's Disease
Scientific title
Study AZ3110866, a Fixed Dose Study of SB-742457 Versus Placebo When Added to Existing Donepezil Treatment in Subjects With Mild-to-moderate Alzheimer's Disease
Secondary ID [1] 0 0
AZ3110866
Universal Trial Number (UTN)
Trial acronym
Linked study record

Health condition
Health condition(s) or problem(s) studied:
Alzheimer's Disease 0 0
Condition category
Condition code
Neurological 0 0 0 0
Alzheimer's disease
Neurological 0 0 0 0
Dementias

Intervention/exposure
Study type
Interventional
Description of intervention(s) / exposure
Treatment: Drugs - SB-742457 15mg
Treatment: Drugs - SB-742457 35mg
Treatment: Drugs - Placebo
Treatment: Drugs - donepezil 5-10mg

Experimental: DONEPEZIL + SB-742457 15 MG - SB-742457 - 15mg added to existing donepezil treatment

Placebo comparator: DONEPEZIL + PLACEBO - Placebo added to existing donepezil

Experimental: DONEPEZIL + SB-742457 35 MG - SB-742457 - 35mg added to existing donepezil


Treatment: Drugs: SB-742457 15mg
SB-742457 - 15mg added to existing donepezil treatment

Treatment: Drugs: SB-742457 35mg
SB-742457 - 35mg added to existing donepezil

Treatment: Drugs: Placebo
Placebo added to existing donepezil

Treatment: Drugs: donepezil 5-10mg
existing donepezil treatment

Intervention code [1] 0 0
Treatment: Drugs
Comparator / control treatment
Control group

Outcomes
Primary outcome [1] 0 0
Change From Baseline in Alzheimer's Disease Assessment Scale - Cognitive Subscale (ADAS-Cog) Total Score at Week 24
Timepoint [1] 0 0
Baseline(Week 0) and Week 24
Primary outcome [2] 0 0
Change From Baseline in Clinical Dementia Rating - Sum of Boxes (CDR-SB) Score at Week 24
Timepoint [2] 0 0
Baseline(Week 0) and Week 24
Secondary outcome [1] 0 0
Change From Baseline in Repeatable Battery for the Assessment of Neuropsychological Status (RBANS) Total Score at Week 24
Timepoint [1] 0 0
Baseline (Week 0) and Week 24
Secondary outcome [2] 0 0
Change From Baseline in ADAS-Cog Total Score at Week 12, 36 and 48
Timepoint [2] 0 0
Baseline (Week 0) and Week 12, 36 and 48
Secondary outcome [3] 0 0
Change From Baseline in CDR-SB Score at Week 12, 36 and 48
Timepoint [3] 0 0
Baseline (Week 0) and Week 12, 36, 48
Secondary outcome [4] 0 0
Change From Baseline in RBANS Score at Week 12, 36 and 48
Timepoint [4] 0 0
Baseline (Week 0) and Week 12, 36 and 48
Secondary outcome [5] 0 0
Change From Baseline in Alzheimer's Disease Co-operative Study Group - Activities of Daily Living Inventory (ADCS- ADL) Total Score at Weeks 12, 24, 36 and 48
Timepoint [5] 0 0
Baseline (Week 0) and Week 12, 24, 36 and 48
Secondary outcome [6] 0 0
Change From Baseline in Mini Mental State Examination (MMSE) Total Score at Week 24 and 48
Timepoint [6] 0 0
Baseline (Week 0) and Week 24 and 48
Secondary outcome [7] 0 0
Number of Participants With Adverse Events (AEs) and Serious Adverse Events (SAEs) During Treatment Phase
Timepoint [7] 0 0
Up to follow-up i.e. 2 weeks post end of treatment (Week 24, Week 48 or Early Withdrawal)
Secondary outcome [8] 0 0
Number of Participants With Parameters of Clinical Concern - Hematology
Timepoint [8] 0 0
Up to Week 48
Secondary outcome [9] 0 0
Number of Participants With Parameters of Clinical Concern - Clinical Chemistry
Timepoint [9] 0 0
Up to Week 48
Secondary outcome [10] 0 0
Exposure Estimates for SB-742457 : Area Under the Concentration Time Curve Over the Dosing Interval at Steady State (AUCtss)
Timepoint [10] 0 0
Post-dose at 3, 8 and 24 hours on Week 0, 1, 3, 6, 12, 18, 24, 30, 36, 42 and 48
Secondary outcome [11] 0 0
Exposure Estimates for SB-742457 : Minimum Concentrations at Steady State (Cmin-ss)
Timepoint [11] 0 0
Post-dose at 3, 8 and 24 hours on Week 0, 1, 3, 6, 12, 18, 24, 30, 36, 42 and 48
Secondary outcome [12] 0 0
Exposure Estimates for Donepezil (Cavgss)
Timepoint [12] 0 0
Post-dose at 12 to 20 hours on Week 0, 1, 3, 6, 12, 18, 24, 30, 36, 42 and 48
Secondary outcome [13] 0 0
Change From Baseline in ADAS-Cog Scale in Participants With APOE4 Gene
Timepoint [13] 0 0
Baseline (Week 0) to Week 24 and Week 48
Secondary outcome [14] 0 0
Change From Baseline in CDR-SB Scale in Participants With APOE4 Gene
Timepoint [14] 0 0
Baseline (Week 0) to Week 24 and Week 48
Secondary outcome [15] 0 0
Change From Baseline in RBANS Scale in Participants With APOE4 Gene
Timepoint [15] 0 0
Baseline (Week 0) to Week 24 and Week 48

Eligibility
Key inclusion criteria
* Subjects and their caregivers must provide informed consent prior to study entry.
* Subjects must have a clinical diagnosis of probable mild-to-moderate Alzheimer's disease with no evidence of disorders that are thought to be the cause of, or contributing to the severity of the subject's dementia and a documented history of at least 6 months of ongoing donepezil therapy with stable dosing for at least the last 2 months.
* Subjects must have a regular caregiver who is willing to attend visits, oversee the subject's compliance with the study and report on the subject's status.
* Female subjects of child-bearing potential must agree to abstinence or an approved form of birth control.
* Subjects must have adequate blood pressure and laboratory values.
Minimum age
50 Years
Maximum age
85 Years
Sex
Both males and females
Can healthy volunteers participate?
No
Key exclusion criteria
* Subjects with a diagnosis of possible, probable or definite vascular dementia may not participate.
* Subjects with known hypersensitivity to sunlight or a history of seizures, previous exposure to SB-742457, taking agents for which there is a theoretical risk of interaction with SB-742457, or taking medication for Alzheimer's disease or centrally acting agents which might impact study outcomes may not participate.

Study design
Purpose of the study
Treatment
Allocation to intervention
Randomised controlled trial
Procedure for enrolling a subject and allocating the treatment (allocation concealment procedures)
Methods used to generate the sequence in which subjects will be randomised (sequence generation)
Masking / blinding
Blinded (masking used)
Who is / are masked / blinded?
The people receiving the treatment/s


The people analysing the results/data
Intervention assignment
Parallel
Other design features
Phase
Phase 2
Type of endpoint/s
Statistical methods / analysis

Recruitment
Recruitment status
Completed
Data analysis
Reason for early stopping/withdrawal
Other reasons
Date of first participant enrolment
Anticipated
Actual
Date of last participant enrolment
Anticipated
Actual
Date of last data collection
Anticipated
Actual
Sample size
Target
Accrual to date
Final
Recruitment in Australia
Recruitment state(s)
NSW,QLD,SA,VIC,WA
Recruitment hospital [1] 0 0
GSK Investigational Site - Kogarah
Recruitment hospital [2] 0 0
GSK Investigational Site - Herston
Recruitment hospital [3] 0 0
GSK Investigational Site - Woodville
Recruitment hospital [4] 0 0
GSK Investigational Site - Ballarat
Recruitment hospital [5] 0 0
GSK Investigational Site - Heidelberg West
Recruitment hospital [6] 0 0
GSK Investigational Site - Kew
Recruitment hospital [7] 0 0
GSK Investigational Site - Nedlands
Recruitment postcode(s) [1] 0 0
2217 - Kogarah
Recruitment postcode(s) [2] 0 0
4029 - Herston
Recruitment postcode(s) [3] 0 0
5011 - Woodville
Recruitment postcode(s) [4] 0 0
3350 - Ballarat
Recruitment postcode(s) [5] 0 0
3084 - Heidelberg West
Recruitment postcode(s) [6] 0 0
3101 - Kew
Recruitment postcode(s) [7] 0 0
6009 - Nedlands
Recruitment outside Australia
Country [1] 0 0
United States of America
State/province [1] 0 0
Arizona
Country [2] 0 0
United States of America
State/province [2] 0 0
California
Country [3] 0 0
United States of America
State/province [3] 0 0
Florida
Country [4] 0 0
United States of America
State/province [4] 0 0
New Jersey
Country [5] 0 0
United States of America
State/province [5] 0 0
New York
Country [6] 0 0
United States of America
State/province [6] 0 0
North Carolina
Country [7] 0 0
United States of America
State/province [7] 0 0
Ohio
Country [8] 0 0
United States of America
State/province [8] 0 0
Oklahoma
Country [9] 0 0
United States of America
State/province [9] 0 0
Tennessee
Country [10] 0 0
United States of America
State/province [10] 0 0
Texas
Country [11] 0 0
United States of America
State/province [11] 0 0
Vermont
Country [12] 0 0
Argentina
State/province [12] 0 0
Buenos Aires
Country [13] 0 0
Argentina
State/province [13] 0 0
Córdova
Country [14] 0 0
Argentina
State/province [14] 0 0
Santa Fe
Country [15] 0 0
Canada
State/province [15] 0 0
New Brunswick
Country [16] 0 0
Canada
State/province [16] 0 0
Nova Scotia
Country [17] 0 0
Canada
State/province [17] 0 0
Ontario
Country [18] 0 0
Canada
State/province [18] 0 0
Quebec
Country [19] 0 0
Canada
State/province [19] 0 0
Québec
Country [20] 0 0
Chile
State/province [20] 0 0
Región Metro De Santiago
Country [21] 0 0
Chile
State/province [21] 0 0
Valparaíso
Country [22] 0 0
Chile
State/province [22] 0 0
Santiago
Country [23] 0 0
Czechia
State/province [23] 0 0
Melnik
Country [24] 0 0
Czechia
State/province [24] 0 0
Olomouc
Country [25] 0 0
Czechia
State/province [25] 0 0
Ostrava
Country [26] 0 0
Czechia
State/province [26] 0 0
Pardubice
Country [27] 0 0
Czechia
State/province [27] 0 0
Plzen
Country [28] 0 0
Czechia
State/province [28] 0 0
Praha 10
Country [29] 0 0
Czechia
State/province [29] 0 0
Praha 1
Country [30] 0 0
Czechia
State/province [30] 0 0
Praha 4
Country [31] 0 0
Germany
State/province [31] 0 0
Baden-Wuerttemberg
Country [32] 0 0
Germany
State/province [32] 0 0
Bayern
Country [33] 0 0
Germany
State/province [33] 0 0
Hessen
Country [34] 0 0
Germany
State/province [34] 0 0
Mecklenburg-Vorpommern
Country [35] 0 0
Germany
State/province [35] 0 0
Niedersachsen
Country [36] 0 0
Germany
State/province [36] 0 0
Nordrhein-Westfalen
Country [37] 0 0
Germany
State/province [37] 0 0
Sachsen
Country [38] 0 0
Germany
State/province [38] 0 0
Thueringen
Country [39] 0 0
Germany
State/province [39] 0 0
Berlin
Country [40] 0 0
Italy
State/province [40] 0 0
Abruzzo
Country [41] 0 0
Italy
State/province [41] 0 0
Campania
Country [42] 0 0
Italy
State/province [42] 0 0
Lazio
Country [43] 0 0
Italy
State/province [43] 0 0
Lombardia
Country [44] 0 0
Italy
State/province [44] 0 0
Piemonte
Country [45] 0 0
Italy
State/province [45] 0 0
Toscana
Country [46] 0 0
Italy
State/province [46] 0 0
Umbria
Country [47] 0 0
Italy
State/province [47] 0 0
Veneto
Country [48] 0 0
Spain
State/province [48] 0 0
Baracaldo/Vizcaya
Country [49] 0 0
Spain
State/province [49] 0 0
Barcelona
Country [50] 0 0
Spain
State/province [50] 0 0
Burgos
Country [51] 0 0
Spain
State/province [51] 0 0
Castellón
Country [52] 0 0
Spain
State/province [52] 0 0
Madrid
Country [53] 0 0
Spain
State/province [53] 0 0
Murcia
Country [54] 0 0
Spain
State/province [54] 0 0
Salamanca
Country [55] 0 0
Spain
State/province [55] 0 0
San Sebastián
Country [56] 0 0
Spain
State/province [56] 0 0
San Vicente Del Raspeig/Alicante
Country [57] 0 0
Spain
State/province [57] 0 0
Valencia

Funding & Sponsors
Primary sponsor type
Commercial sector/industry
Name
GlaxoSmithKline
Address
Country

Ethics approval
Ethics application status

Summary
Brief summary
Trial website
Trial related presentations / publications
Public notes

Contacts
Principal investigator
Name 0 0
GSK Clinical Trials
Address 0 0
GlaxoSmithKline
Country 0 0
Phone 0 0
Fax 0 0
Email 0 0
Contact person for public queries
Name 0 0
Address 0 0
Country 0 0
Phone 0 0
Fax 0 0
Email 0 0
Contact person for scientific queries

No information has been provided regarding IPD availability


What supporting documents are/will be available?

No Supporting Document Provided



Results publications and other study-related documents

No documents have been uploaded by study researchers.